Pyrene Actin

 
Pyrene Actin
Actin polymerization kinetics
Cys374-labeled G-actin
100% and 10% pyrene formats
 
Fluorometric analysis of pyrene-actin polymerization and depolymerization kinetics
Actin protein cube
Fluorometric kinetic readout
Pyrene-actin fluorescence reports actin polymerization, depolymerization and ligand-dependent filament dynamics.
Fast and reliable analysis of actin dynamics

Pyrene Actin for quantitative polymerization assays

Fluorescent Cys374-labeled G-actin for sensitive fluorometric analysis of actin assembly, disassembly, nucleation and ligand-dependent filament dynamics.

Pyrene Actin from Hypermol® is chemically modified G-actin carrying a fluorescent pyrenyl group covalently attached to Cys374 at the C-terminus of actin. Upon polymerization, pyrene fluorescence provides a robust kinetic signal for monitoring actin filament formation and turnover.

Pyrene-actin assays are widely used to characterize actin-binding proteins, myosins, drugs, natural compounds and other ligands that modulate polymerization, depolymerization or nucleation. Hypermol® provides defined 100% and 10% pyrene-actin formats with high polymerization competence and instant solubility.

Kinetics
Real-time fluorometric monitoring of polymerization and depolymerization.
Defined labeling
1:1 pyrene:actin ratio for 100% pyrene actin; 1:10 for 10% pyrene actin.
Assay ready
Highly polymerizable, instantly soluble actin for reproducible pyrene assays.
Browse Pyrene Actin
Typical applications
Fluorometry, fluorimetry, pyrene-actin assays, polymerization kinetics, depolymerization kinetics, nucleation assays and ligand-dependent actin dynamics.
Product focus
Pyrene-labeled actin at defined dye/protein ratios for sensitive, quantitative and reproducible analysis of actin filament dynamics.
Hypermol Satisfaction Guarantee
Validated product quality with Satisfaction Guarantee.
Proteins from Hypermol® are of validated high biological activity, as described in our publications.
   
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Introduction to Fluorometry is Actin
Pyrene Actin to measure actin polymerisation and depolymerisation


G-actin (globular actin) is a monomeric protein, which is the subunit of the actin microfilaments. Since G-actin polymerizes reversibly into double-helical microfilaments (the "actin helix"), it constitutes the "actin-based cytoskeleton" of  practically all eucaryotic cells. Actin became a key player for cellular movement and force exercise (muscle, cell division). This arose only by the ability of hundreds of proteins with highly indidviual capabilities to evolve binding sites for actin and thus to utilize the actin filaments to assemble, and disassemble multi-protein-complex suprastructures needed for the motile and scaffolding functions of living cells.

To characterize actin-binding proteins, but also drugs / natural compounds / non-protein ligands in their abilty to modify the polymerization or depolymerization of actin, the actin kinetics are measured by fluorometry. This method requires Pyrene-Actin, which is chemically modified G-actin, carrying a pyrenyl group covalently bound to Cys374 at the C-term of the molecule.

The actin polymerization can be induced simply by mono- or divalent cations  (in-vitro conditions). and the actin kinetic can then be measured fluorometrically. Upon excitation a characteristic kinetic is observed, which  instantly shows the effect of ligands on the assembly or disassembly of the actin filaments.